Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6057 |
URMC-099
|
ROCK; MLK; VEGFR; SGK; DNA Alkylation; Trk receptor; c-Met/HGFR; LRRK2; MEK; IGF-1R; Syk; Bcr-Abl; CDK; Src; Aurora Kinase; Autophagy | Angiogenesis; Autophagy; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; MAPK; Metabolism; Stem Cells; Tyrosine Kinase/Adaptors |
URMC-099 是一种具有优异的血脑屏障穿透性的,可口服的混合谱系激酶 3 抑制剂,IC50为14 nM。 |